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1FD0

ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE RARGAMMA-SELECTIVE RETINOID SR11254

Summary for 1FD0
Entry DOI10.2210/pdb1fd0/pdb
Related1EXA 1EXX 1fcx 1fcy 1fcz 2LBD 3LBD
DescriptorRETINOIC ACID RECEPTOR GAMMA-1, 6-[HYDROXYIMINO-(5,5,8,8-TETRAMETHYL-5,6,7,8-TETRAHYDRO-NAPHTALEN-2-YL)-METHYL]-NAPHTALENE-2-CARBOXYLIC ACID, DODECYL-ALPHA-D-MALTOSIDE, ... (4 entities in total)
Functional Keywordsisotype selectivity, retinoid ligand complexes, drug design, antiparallel alpha-helical sandwich fold, ch...o hydrogen bond, structural proteomics in europe, spine, structural genomics, gene regulation
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight27447.18
Authors
Klaholz, B.P.,Moras, D.,Structural Proteomics in Europe (SPINE) (deposition date: 2000-07-19, release date: 2002-09-27, Last modification date: 2023-08-09)
Primary citationKlaholz, B.,Moras, D.
C-H...O hydrogen bonds in the nuclear receptor RARgamma--a potential tool for drug selectivity.
Structure, 10:1197-1204, 2002
Cited by
PubMed: 12220491
DOI: 10.1016/S0969-2126(02)00828-6
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.38 Å)
Structure validation

217705

건을2024-03-27부터공개중

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