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1FD0

ISOTYPE SELECTIVITY OF THE HUMAN RETINOIC ACID NUCLEAR RECEPTOR HRAR: THE COMPLEX WITH THE RARGAMMA-SELECTIVE RETINOID SR11254

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0048384biological_processretinoic acid receptor signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 254 A 450
ChainResidue
APHE201
ASER289
AGLY303
APHE304
ALEU400
AILE412
AHOH549
APHE230
AALA234
ACYS237
ALEU271
AMET272
AILE275
AARG278
APHE288

site_idAC2
Number of Residues18
DetailsBINDING SITE FOR RESIDUE LMU A 451
ChainResidue
ALYS240
AGLU243
ALEU263
ACYS267
AASP340
AGLN354
APRO377
ALEU380
AILE383
ATHR384
AARG387
AMET415
AHOH561
AHOH607
AHOH648
AHOH688
AHOH747
AHOH782

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS401

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PDB entries from 2024-09-11

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