1X7E
CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA COMPLEXED WITH WAY-244
Summary for 1X7E
Entry DOI | 10.2210/pdb1x7e/pdb |
Related | 1U3Q 1U3R 1U3S 1U9E 1X76 1X78 1X7B 1X7D 1X7J 1X7R |
Descriptor | Estrogen receptor 1 (alpha), steroid receptor coactivator-3, [5-HYDROXY-2-(4-HYDROXYPHENYL)-1-BENZOFURAN-7-YL]ACETONITRILE, ... (4 entities in total) |
Functional Keywords | estrogen receptor, estrogen receptor beta, er-beta, er, estrogen receptor alpha, er-alpha, estrogen, nuclear recept transcription factor, agonist, transcription |
Biological source | Homo sapiens (human) More |
Cellular location | Isoform 1: Nucleus. Isoform 3: Nucleus: P03372 |
Total number of polymer chains | 4 |
Total formula weight | 59818.49 |
Authors | Manas, E.S.,Unwalla, R.J.,Xu, Z.B.,Malamas, M.S.,Miller, C.P.,Harris, H.A.,Hsiao, C.,Akopian, T.,Hum, W.T.,Malakian, K.,Wolfrom, S.,Bapat, A.,Bhat, R.A.,Stahl, M.L.,Somers, W.S.,Alvarez, J.C. (deposition date: 2004-08-13, release date: 2005-03-01, Last modification date: 2024-04-03) |
Primary citation | Manas, E.S.,Unwalla, R.J.,Xu, Z.B.,Malamas, M.S.,Miller, C.P.,Harris, H.A.,Hsiao, C.,Akopian, T.,Hum, W.T.,Malakian, K.,Wolfrom, S.,Bapat, A.,Bhat, R.A.,Stahl, M.L.,Somers, W.S.,Alvarez, J.C. Structure-Based Design of Estrogen Receptor-Beta Selective Ligands J.Am.Chem.Soc., 126:15106-15119, 2004 Cited by PubMed: 15548008DOI: 10.1021/ja047633o PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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