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1X7B

CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR BETA COMPLEXED WITH ERB-041

Summary for 1X7B
Entry DOI10.2210/pdb1x7b/pdb
Related1U3Q 1U3R 1U3S 1U9E 1X76 1X78 1X7J 1X7R
DescriptorEstrogen receptor beta, STEROID RECEPTOR COACTIVATOR-1, 2-(3-FLUORO-4-HYDROXYPHENYL)-7-VINYL-1,3-BENZOXAZOL-5-OL, ... (4 entities in total)
Functional Keywordsestrogen receptor, estrogen receptor beta, er-beta, er, estrogen, nuclear receptor, transcription factor, agonist, transcription
Biological sourceHomo sapiens (human)
More
Cellular locationNucleus: Q92731
Total number of polymer chains4
Total formula weight57533.96
Authors
Primary citationManas, E.S.,Unwalla, R.J.,Xu, Z.B.,Malamas, M.S.,Miller, C.P.,Harris, H.A.,Hsiao, C.,Akopian, T.,Hum, W.T.,Malakian, K.,Wolfrom, S.,Bapat, A.,Bhat, R.A.,Stahl, M.L.,Somers, W.S.,Alvarez, J.C.
Structure-Based Design of Estrogen Receptor-Beta Selective Ligands
J.Am.Chem.Soc., 126:15106-15119, 2004
Cited by
PubMed: 15548008
DOI: 10.1021/ja047633o
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

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