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9H32

T2R-TTL-PROTAC3 complex

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, C
(A, C)
Tubulin alpha-1B chainpolymer45150204.42UniProt (P81947)Bos taurus (domestic cattle)Alpha-tubulin ubiquitous,Tubulin K-alpha-1,Tubulin alpha-ubiquitous chain
2B, D
(B, D)
Tubulin beta-2B chainpolymer44549999.92UniProt (Q6B856)Bos taurus (domestic cattle)
3E
(E)
Stathmin-4polymer14316844.21UniProt (P63043)Rattus norvegicus (Norway rat)Stathmin-like protein B3,RB3
4F
(F)
Tubulin--tyrosine ligasepolymer38444378.51UniProt (A0A8V0Z8P0)Gallus gallus (chicken)
5G, N
(A, C)
GUANOSINE-5'-TRIPHOSPHATEnon-polymer523.22Chemie (GTP)
6H, K, O, R, V
(A, B, C, D, F)
MAGNESIUM IONnon-polymer24.35Chemie (MG)
7I, L, P, T
(A, B, C, E)
CALCIUM IONnon-polymer40.14Chemie (CA)
8J, Q
(B, D)
GUANOSINE-5'-DIPHOSPHATEnon-polymer443.22Chemie (GDP)
9M
(B)
2-(N-MORPHOLINO)-ETHANESULFONIC ACIDnon-polymer195.21Chemie (MES)
10S
(D)
(1S,2R,3S,5S,6S,16E,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.1~10,14~.0~3,5~]hexacosa-10(26),11,13,16-tetraen-6-yl 4-(2-{4-[4-({2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-2,3-dihydro-1H-isoindol-4-yl}amino)-4-oxobutyl]-1H-1,2,3-triazol-1-yl}ethyl)benzoatenon-polymer1093.61Chemie (A1ISD)
11U
(F)
PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTERnon-polymer505.21Chemie (ACP)
12AA, BA, W, X, Y...
(E, F, A, B, C...)
waterwater18.0282Chemie (HOH)
Sequence modifications
E: 5 - 145 (UniProt: P63043)
PDBExternal DatabaseDetails
Met 3-initiating methionine
Ala 4-expression tag
F: 1 - 52 (UniProt: A0A8V0Z8P0)
F: 53 - 378 (UniProt: A0A8V0Z8P0)
PDBExternal DatabaseDetails
His 379-expression tag
His 380-expression tag
His 381-expression tag
His 382-expression tag
His 383-expression tag
His 384-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains6
Total formula weight261631.3
Non-Polymers*Number of molecules16
Total formula weight4008.7
All*Total formula weight265640.0
*Water molecules are not included.

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PDB entries from 2025-10-29

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