8X63
CryoEM structure of the histamine H1 receptor-BRIL/Anti BRIL Fab complex with mepyramine
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | B | Histamine H1 receptor,Soluble cytochrome b562 | polymer | 438 | 50629.4 | 1 | UniProt (P35367) UniProt (P0ABE7) Pfam (PF00001) Pfam (PF07361) In PDB | Homo sapiens (human) | H1R,HH1R,Cytochrome b-562 |
2 | B | mepyramine | non-polymer | 285.4 | 1 | Chemie (Y5E) |
Sequence modifications
B: 20 - 217 (UniProt: P35367)
B: 408 - 483 (UniProt: P35367)
B: 306 - 348 (UniProt: P0ABE7)
B: 353 - 403 (UniProt: P0ABE7)
PDB | External Database | Details |
---|---|---|
Asp 12 | - | expression tag |
Tyr 13 | - | expression tag |
Lys 14 | - | expression tag |
Asp 15 | - | expression tag |
Asp 16 | - | expression tag |
Asp 17 | - | expression tag |
Asp 18 | - | expression tag |
Lys 19 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Lys 218 | - | linker |
Arg 219 | - | linker |
Gln 220 | - | linker |
Leu 221 | - | linker |
Lys 484 | - | expression tag |
Ile 485 | - | expression tag |
Ala 486 | - | expression tag |
Ala 487 | - | expression tag |
Leu 488 | - | expression tag |
Lys 489 | - | expression tag |
Glu 490 | - | expression tag |
Lys 491 | - | expression tag |
Ile 492 | - | expression tag |
Ala 493 | - | expression tag |
Ala 494 | - | expression tag |
Leu 495 | - | expression tag |
Lys 496 | - | expression tag |
Glu 497 | - | expression tag |
Lys 498 | - | expression tag |
Ile 499 | - | expression tag |
Ala 500 | - | expression tag |
Ala 501 | - | expression tag |
Leu 502 | - | expression tag |
Lys 503 | - | expression tag |
Glu 504 | - | expression tag |
Ala 505 | - | expression tag |
Glu 506 | - | expression tag |
Glu 507 | - | expression tag |
Lys 508 | - | expression tag |
Arg 509 | - | expression tag |
Ala 510 | - | expression tag |
Ser 511 | - | expression tag |
Arg 512 | - | expression tag |
Leu 513 | - | expression tag |
Glu 514 | - | expression tag |
Glu 515 | - | expression tag |
Glu 516 | - | expression tag |
Leu 517 | - | expression tag |
Arg 518 | - | expression tag |
Arg 519 | - | expression tag |
Arg 520 | - | expression tag |
Leu 521 | - | expression tag |
Thr 522 | - | expression tag |
Glu 523 | - | expression tag |
Gly 524 | - | expression tag |
Ser 525 | - | expression tag |
His 526 | - | expression tag |
His 527 | - | expression tag |
His 528 | - | expression tag |
His 529 | - | expression tag |
His 530 | - | expression tag |
His 531 | - | expression tag |
His 532 | - | expression tag |
His 533 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Trp 312 | Met 29 | engineered mutation |
PDB | External Database | Details |
---|---|---|
Ser 349 | - | linker |
Gly 350 | - | linker |
Ser 351 | - | linker |
Gly 352 | - | linker |
Ile 400 | His 124 | engineered mutation |
Leu 404 | - | linker |
Lys 405 | - | linker |
Phe 406 | - | linker |
Cys 407 | - | linker |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 1 |
Total formula weight | 50629.4 | |
Non-Polymers* | Number of molecules | 1 |
Total formula weight | 285.4 | |
All* | Total formula weight | 50914.7 |