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8PYI

Human IGF1R with inhibitor 6

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B, C, D, E...
(AAA, BBB, CCC, DDD, EEE...)
Insulin-like growth factor 1 receptor beta chainpolymer32136716.08UniProt (P08069)
Pfam (PF07714)
Homo sapiens (human)
2I, J, K, L, M...
(AAA, BBB, CCC, DDD, EEE...)
3-[8-azanyl-1-(4-ethoxy-8-fluoranyl-2-phenyl-quinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutan-1-olnon-polymer483.58Chemie (IER)
3Q, R, S, T, U...
(AAA, BBB, CCC, DDD, EEE...)
waterwater18.0174Chemie (HOH)
Sequence modifications
AAA, BBB, CCC, DDD, EEE, FFF, GGG, HHH: 974 - 1286 (UniProt: P08069)
PDBExternal DatabaseDetails
Met 973-initiating methionine
Ala 1287-expression tag
Glu 1288-expression tag
Asn 1289-expression tag
Leu 1290-expression tag
Tyr 1291-expression tag
Phe 1292-expression tag
Gln 1293-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains8
Total formula weight293727.9
Non-Polymers*Number of molecules8
Total formula weight3868.3
All*Total formula weight297596.2
*Water molecules are not included.

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PDB entries from 2025-07-23

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