8G0H
Human PARP1 deltaV687-E688 bound to UKTT5 (compound 10) and to a DNA double strand break.
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | O, N | DNA (5'-D(*CP*GP*AP*CP*G)-3') | polymer | 5 | 1505.0 | 2 | DNA molecule | ||
2 | P, M | DNA (5'-D(*CP*GP*TP*CP*G)-3') | polymer | 5 | 1496.0 | 2 | DNA molecule | ||
3 | D, B | Poly [ADP-ribose] polymerase 1 | polymer | 504 | 56909.9 | 2 | UniProt (P09874) Pfam (PF05406) Pfam (PF02877) Pfam (PF00644) In PDB | Homo sapiens (human) | PARP-1,ADP-ribosyltransferase diphtheria toxin-like 1,ARTD1,DNA ADP-ribosyltransferase PARP1,NAD(+) ADP-ribosyltransferase 1,ADPRT 1,Poly[ADP-ribose] synthase 1,Protein poly-ADP-ribosyltransferase PARP1 |
4 | A, C | Fusion of human PARP1 zinc fingers 1 and 3 (Zn1, Zn3),Poly [ADP-ribose] polymerase 1 | polymer | 276 | 31262.8 | 2 | UniProt (P09874) Pfam (PF00645) Pfam (PF21728) Pfam (PF08063) In PDB | Homo sapiens (human) | PARP-1,ADP-ribosyltransferase diphtheria toxin-like 1,ARTD1,DNA ADP-ribosyltransferase PARP1,NAD(+) ADP-ribosyltransferase 1,ADPRT 1,Poly[ADP-ribose] synthase 1,Protein poly-ADP-ribosyltransferase PARP1 |
5 | D, B | 2-(4-{[2-(1H-benzimidazol-2-yl)ethyl]carbamoyl}phenyl)-1H-benzimidazole-7-carboxamide | non-polymer | 424.5 | 2 | Chemie (YH0) | |||
6 | A, C | ZINC ION | non-polymer | 65.4 | 4 | Chemie (ZN) |
Sequence modifications
D, B: 518 - 1014 (UniProt: P09874)
A, C: 1 - 205 (UniProt: P09874)
A, C: 206 - 366 (UniProt: P09874)
PDB | External Database | Details |
---|---|---|
Met 517 | - | initiating methionine |
- | Val 687 | deletion |
- | Glu 688 | deletion |
Ala 762 | Val 762 | variant |
Leu 1015 | - | expression tag |
Glu 1016 | - | expression tag |
His 1017 | - | expression tag |
His 1018 | - | expression tag |
His 1019 | - | expression tag |
His 1020 | - | expression tag |
His 1021 | - | expression tag |
His 1022 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Met -19 | - | expression tag |
Gly -18 | - | expression tag |
Ser -17 | - | expression tag |
Ser -16 | - | expression tag |
His -15 | - | expression tag |
His -14 | - | expression tag |
His -13 | - | expression tag |
His -12 | - | expression tag |
His -11 | - | expression tag |
His -10 | - | expression tag |
Ser -9 | - | expression tag |
Ser -8 | - | expression tag |
Gly -7 | - | expression tag |
Leu -6 | - | expression tag |
Val -5 | - | expression tag |
Pro -4 | - | expression tag |
Arg -3 | - | expression tag |
Gly -2 | - | expression tag |
Ser -1 | - | expression tag |
His 0 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 8 |
Total formula weight | 182347.6 | |
Non-Polymers* | Number of molecules | 6 |
Total formula weight | 1110.5 | |
All* | Total formula weight | 183458.1 |