7XWO
Neurokinin A bound to active human neurokinin 2 receptor in complex with G324
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | B | Soluble cytochrome b562,Substance-K receptor | polymer | 505 | 57108.2 | 1 | UniProt (P0ABE7) UniProt (P21452) Pfam (PF07361) Pfam (PF00001) In PDB | Homo sapiens (human) | Cytochrome b-562,SKR,NK-2 receptor,NK-2R,Neurokinin A receptor,Tachykinin receptor 2 |
2 | C | Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 | polymer | 344 | 37784.3 | 1 | UniProt (P54311) Pfam (PF00400) In PDB | Rattus norvegicus (Norway rat) | Transducin beta chain 1 |
3 | E | scFv | polymer | 304 | 32692.5 | 1 | Rattus norvegicus | ||
4 | F | G324 | polymer | 361 | 41710.3 | 1 | Homo sapiens | ||
5 | G | Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 | polymer | 71 | 7861.1 | 1 | UniProt (P63212) Pfam (PF00631) In PDB | Bos taurus (cattle) | G gamma-I |
6 | D | HIS-LYS-THR-ASP-SER-PHE-VAL-GLY-LEU-MET-NH2 | polymer | 11 | 1207.4 | 1 | UniProt (by SIFTS) (P20366) In PDB | Homo sapiens |
Sequence modifications
B: -105 - -1 (UniProt: P0ABE7)
B: 1 - 345 (UniProt: P21452)
C: 7 - 345 (UniProt: P54311)
PDB | External Database | Details |
---|---|---|
Met -153 | - | initiating methionine |
Lys -152 | - | expression tag |
Thr -151 | - | expression tag |
Ile -150 | - | expression tag |
Ile -149 | - | expression tag |
Ala -148 | - | expression tag |
Leu -147 | - | expression tag |
Ser -146 | - | expression tag |
Tyr -145 | - | expression tag |
Ile -144 | - | expression tag |
Phe -143 | - | expression tag |
Cys -142 | - | expression tag |
Leu -141 | - | expression tag |
Val -140 | - | expression tag |
Phe -139 | - | expression tag |
Ala -138 | - | expression tag |
Asp -137 | - | expression tag |
Tyr -136 | - | expression tag |
Lys -135 | - | expression tag |
Asp -134 | - | expression tag |
Asp -133 | - | expression tag |
Asp -132 | - | expression tag |
Asp -131 | - | expression tag |
Ala -130 | - | expression tag |
Lys -129 | - | expression tag |
Leu -128 | - | expression tag |
Gln -127 | - | expression tag |
Thr -126 | - | expression tag |
Met -125 | - | expression tag |
His -124 | - | expression tag |
His -123 | - | expression tag |
His -122 | - | expression tag |
His -121 | - | expression tag |
His -120 | - | expression tag |
His -119 | - | expression tag |
His -118 | - | expression tag |
His -117 | - | expression tag |
His -116 | - | expression tag |
His -115 | - | expression tag |
Glu -114 | - | expression tag |
Asn -113 | - | expression tag |
Leu -112 | - | expression tag |
Tyr -111 | - | expression tag |
Phe -110 | - | expression tag |
Gln -109 | - | expression tag |
Gly -108 | - | expression tag |
Gly -107 | - | expression tag |
Thr -106 | - | expression tag |
Trp -99 | Met 29 | conflict |
Ile -4 | His 124 | conflict |
Leu 0 | - | linker |
PDB | External Database | Details |
---|---|---|
Lys 346 | - | expression tag |
Leu 347 | - | expression tag |
Val 348 | - | expression tag |
Glu 349 | - | expression tag |
Lys 350 | - | expression tag |
Tyr 351 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Gly 2 | - | expression tag |
Ser 3 | - | expression tag |
Leu 4 | - | expression tag |
Leu 5 | - | expression tag |
Gln 6 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 6 |
Total formula weight | 178363.8 | |
All* | Total formula weight | 178363.8 |