7UL2
CryoEM Structure of Inactive NTSR1 Bound to SR48692 and Nb6
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | R | Neurotensin receptor 1 | polymer | 419 | 47084.4 | 1 | UniProt (P30989) UniProt (P41145) Pfam (PF00001) In PDB | Homo sapiens (human) | NT-R-1,NTR1,High-affinity levocabastine-insensitive neurotensin receptor,NTRH,K-OR-1,KOR-1 |
2 | D | Nanobody 6 | polymer | 133 | 14730.3 | 1 | Lama glama | ||
3 | R | 2-[[1-(7-chloranylquinolin-4-yl)-5-(2,6-dimethoxyphenyl)pyrazol-3-yl]carbonylamino]adamantane-2-carboxylic acid | non-polymer | 587.1 | 1 | Chemie (Q6Q) | |||
4 | R | SODIUM ION | non-polymer | 23.0 | 1 | Chemie (NA) | |||
5 | water | water | 18.0 | 13 | Chemie (HOH) |
Sequence modifications
R: 20 - 255 (UniProt: P30989)
R: 256 - 308 (UniProt: P41145)
R: 309 - 418 (UniProt: P30989)
PDB | External Database | Details |
---|---|---|
Asp -19 | - | expression tag |
Tyr -18 | - | expression tag |
Lys -17 | - | expression tag |
Asp -16 | - | expression tag |
Asp -15 | - | expression tag |
Asp -14 | - | expression tag |
Asp -13 | - | expression tag |
Ala -12 | - | expression tag |
Met -11 | - | expression tag |
Gly -10 | - | expression tag |
Gln -9 | - | expression tag |
Pro -8 | - | expression tag |
Gly -7 | - | expression tag |
Asn -6 | - | expression tag |
Gly -5 | - | expression tag |
Ser -4 | - | expression tag |
Ala -3 | - | expression tag |
Phe -2 | - | expression tag |
Leu -1 | - | expression tag |
Leu 0 | - | expression tag |
Ala 1 | - | expression tag |
Pro 2 | - | expression tag |
Asn 3 | - | expression tag |
Arg 4 | - | expression tag |
Ser 5 | - | expression tag |
His 6 | - | expression tag |
Ala 7 | - | expression tag |
Pro 8 | - | expression tag |
Asp 9 | - | expression tag |
His 10 | - | expression tag |
Asp 11 | - | expression tag |
Val 12 | - | expression tag |
Glu 13 | - | expression tag |
Asn 14 | - | expression tag |
Leu 15 | - | expression tag |
Tyr 16 | - | expression tag |
Phe 17 | - | expression tag |
Gln 18 | - | expression tag |
Gly 19 | - | expression tag |
Leu 85 | Ala 85 | conflict |
PDB | External Database | Details |
---|---|---|
Ala 307 | Val 278 | conflict |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 61814.6 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 610.1 | |
All* | Total formula weight | 62424.7 |