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7JIU

HUMAN PI3KDELTA IN COMPLEX WITH COMPOUND 2F

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1APhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformpolymer946110084.21UniProt (P42336)
Pfam (PF00794)
Pfam (PF00792)
Pfam (PF00613)
Pfam (PF00454)
In PDB
Homo sapiensPtdIns-3-kinase subunit alpha,Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit alpha,p110alpha,Phosphoinositide-3-kinase catalytic alpha polypeptide,Serine/threonine protein kinase PIK3CA
2A(3S)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9H-purin-6-yl]-3-methyl-1,3-dihydro-2H-indol-2-onenon-polymer475.51Chemie (VBS)
3waterwater18.0289Chemie (HOH)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight110084.2
Non-Polymers*Number of molecules1
Total formula weight475.5
All*Total formula weight110559.7
*Water molecules are not included.

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PDB entries from 2024-06-12

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