7EZC
Adenosine A2a receptor mutant-I92N
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, B | Adenosine receptor A2a,Soluble cytochrome b562 | polymer | 431 | 48158.9 | 2 | UniProt (P29274) UniProt (P0ABE7) Pfam (PF00001) Pfam (PF07361) In PDB | Homo sapiens (human) | Cytochrome b-562 |
2 | A, B | 6-(2,2-diphenylethylamino)-9-[(2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-oxolan-2-yl]-N-[2-[(1-pyridin-2-ylpiperidin-4-yl)carbamoylamino]ethyl]purine-2-carboxamide | non-polymer | 777.9 | 2 | Chemie (UKA) |
Sequence modifications
A, B: 2 - 208 (UniProt: P29274)
A, B: 1001 - 1101 (UniProt: P0ABE7)
A, B: 219 - 308 (UniProt: P29274)
PDB | External Database | Details |
---|---|---|
Asp -8 | - | expression tag |
Tyr -7 | - | expression tag |
Lys -6 | - | expression tag |
Asp -5 | - | expression tag |
Asp -4 | - | expression tag |
Asp -3 | - | expression tag |
Asp -2 | - | expression tag |
Gly -1 | - | expression tag |
Ala 0 | - | expression tag |
Pro 1 | - | expression tag |
Asn 92 | Ile 92 | engineered mutation |
PDB | External Database | Details |
---|---|---|
Trp 1007 | Met 29 | engineered mutation |
Ile 1102 | - | linker |
Gln 1103 | - | linker |
Lys 1104 | - | linker |
Tyr 1105 | - | linker |
Leu 1106 | - | linker |
PDB | External Database | Details |
---|---|---|
Arg 309 | - | expression tag |
Gln 310 | - | expression tag |
Gln 311 | - | expression tag |
Glu 312 | - | expression tag |
Pro 313 | - | expression tag |
Phe 314 | - | expression tag |
Lys 315 | - | expression tag |
Ala 316 | - | expression tag |
His 317 | - | expression tag |
His 318 | - | expression tag |
His 319 | - | expression tag |
His 320 | - | expression tag |
His 321 | - | expression tag |
His 322 | - | expression tag |
His 323 | - | expression tag |
His 324 | - | expression tag |
His 325 | - | expression tag |
His 326 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 96317.9 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 1555.7 | |
All* | Total formula weight | 97873.6 |