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3FAT

X-ray structure of iGluR4 flip ligand-binding core (S1S2) in complex with (S)-AMPA at 1.90A resolution

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B, C
(A, B, C)
Glutamate receptor 4polymer26029020.53UniProt (P19493)
Pfam (PF10613)
Pfam (PF00060)
Rattus norvegicus (rat)ionotropic glutamate receptor 4, GluR-4, GluR4, GluR-D, Glutamate receptor ionotropic, AMPA 4, AMPA-selective glutamate receptor 4
2D, K, T
(A, B, C)
(S)-ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACIDnon-polymer186.23Chemie (AMQ)
3E, F, G, H, L...
(A, B, C)
SULFATE IONnon-polymer96.17Chemie (SO4)
4I, M, N, O, P...
(A, B, C)
GLYCEROLnon-polymer92.19Chemie (GOL)
5AA, BA, J, Q, R...
(C, A, B)
ACETIC ACIDnon-polymer60.16Chemie (ACY)
6CA, DA, EA
(A, B, C)
waterwater18.0630Chemie (HOH)
Sequence modifications
A, B, C: 2 - 115 (UniProt: P19493)
PDBExternal DatabaseDetails
Gly 1-expression tag
A, B, C: 118 - 260 (UniProt: P19493)
PDBExternal DatabaseDetails
Gly 116-linker
Thr 117-linker
Ile 198Thr 734SEE REMARK 999
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains3
Total formula weight87061.6
Non-Polymers*Number of molecules25
Total formula weight2420.1
All*Total formula weight89481.7
*Water molecules are not included.

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PDB entries from 2025-06-18

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