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1C8K

FLAVOPIRIDOL INHIBITS GLYCOGEN PHOSPHORYLASE BY BINDING AT THE INHIBITOR SITE

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
PROTEIN (GLYCOGEN PHOSPHORYLASE)polymer84297291.21UniProt (P00489)
Pfam (PF00343)
Oryctolagus cuniculus (rabbit)
2B
(A)
PYRIDOXAL-5'-PHOSPHATEnon-polymer247.11Chemie (PLP)
3C
(A)
2-(2-CHLORO-PHENYL)-5,7-DIHYDROXY-8-(3-HYDROXY-1-METHYL-PIPERIDIN-4-YL)-4H-BENZOPYRAN-4-ONEnon-polymer401.81Chemie (CPB)
4D
(A)
waterwater18.0331Chemie (HOH)
Sequence modifications
A: 1 - 842 (UniProt: P00489)
PDBExternal DatabaseDetails
Ile 380Leu 380conflict
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight97291.2
Non-Polymers*Number of molecules2
Total formula weight649.0
All*Total formula weight97940.2
*Water molecules are not included.

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PDB entries from 2025-06-11

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