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4R1V

Identification and optimization of pyridazinones as potent and selective c-Met kinase inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF4r1v.cif.gz Display(147.57 KB)
4r1v.cif
PDBx/mmJSONall4r1v.json.gz Display (Tree)(106.73 KB)
4r1v.json
no-atom4r1v-noatom.json.gz Display (Header)(14.80 KB)
4r1v-noatom.json
add only4r1v-plus.json.gz Display(1.20 KB)
4r1v-plus.json
PDBMLall4r1v.xml.gz Display(203.56 KB)
4r1v.xml
no-atom4r1v-noatom.xml.gz Display(27.67 KB)
4r1v-noatom.xml
ext-atom4r1v-extatom.xml.gz Display(62.58 KB)
4r1v-extatom.xml
PDBpdb4r1v.ent.gz Display(115.46 KB)
pdb4r1v.ent
RDF4r1v.rdf.gz Visualize(79.09 KB)
4r1v.rdf
Structure factorsr4r1vsf.ent.gz Display(1.20 MB)
r4r1vsf.ent
Biological unit (mmCIF format)4r1v-assembly1.cif.gz Display(139.16 KB)
4r1v-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4r1v.pdb1.gz Display(110.24 KB)
4r1v.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4r1v_validation.pdf.gz Display(724.93 KB)
4r1v_validation.pdf
PDF-full4r1v_full_validation.pdf.gz Display(726.60 KB)
4r1v_full_validation.pdf
mmCIF4r1v_validation.cif.gz Display(25.30 KB)
4r1v_validation.cif
XML4r1v_validation.xml.gz Display(16.45 KB)
4r1v_validation.xml
PNG4r1v_multipercentile_validation.png.gz Display(168.77 KB)
4r1v_multipercentile_validation.png
SVG4r1v_multipercentile_validation.svg.gz Display(946.00 B)
4r1v_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4r1v_validation_2fo-fc_map_coef.cif.gz Display(1.21 MB)
4r1v_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4r1v_validation_fo-fc_map_coef.cif.gz Display(1.20 MB)
4r1v_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4r1v_validation_2fo-fc_map_coef.mtz Visualize(1.96 MB)
fo-fc (MTZ)4r1v_validation_fo-fc_map_coef.mtz Visualize(1.96 MB)

222415

PDB entries from 2024-07-10

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