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4P1R

Crystal Structure of PDE10A with Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF4p1r.cif.gz Display(165.22 KB)
4p1r.cif
PDBx/mmJSONall4p1r.json.gz Display (Tree)(110.59 KB)
4p1r.json
no-atom4p1r-noatom.json.gz Display (Header)(21.91 KB)
4p1r-noatom.json
add only4p1r-plus.json.gz Display(1000.00 B)
4p1r-plus.json
PDBMLall4p1r.xml.gz Display(223.40 KB)
4p1r.xml
no-atom4p1r-noatom.xml.gz Display(45.41 KB)
4p1r-noatom.xml
ext-atom4p1r-extatom.xml.gz Display(134.75 KB)
4p1r-extatom.xml
PDBpdb4p1r.ent.gz Display(128.23 KB)
pdb4p1r.ent
RDF4p1r.rdf.gz Visualize(119.19 KB)
4p1r.rdf
Structure factorsr4p1rsf.ent.gz Display(1.14 MB)
r4p1rsf.ent
Biological unit (mmCIF format)4p1r-assembly1.cif.gz Display(226.56 KB)
4p1r-assembly1.cif (A)

*software defined assembly, 3 molecule(s) (trimeric)

4p1r-assembly2.cif.gz Display(217.98 KB)
4p1r-assembly2.cif (B)

*software defined assembly, 3 molecule(s) (trimeric)

Biological unit (PDB format)4p1r.pdb1.gz Display(182.32 KB)
4p1r.pdb1 (A)

*software defined assembly, 3 molecule(s) (trimeric)

4p1r.pdb2.gz Display(175.38 KB)
4p1r.pdb2 (B)

*software defined assembly, 3 molecule(s) (trimeric)

Validation reportsPDF4p1r_validation.pdf.gz Display(929.97 KB)
4p1r_validation.pdf
PDF-full4p1r_full_validation.pdf.gz Display(939.00 KB)
4p1r_full_validation.pdf
mmCIF4p1r_validation.cif.gz Display(50.34 KB)
4p1r_validation.cif
XML4p1r_validation.xml.gz Display(33.81 KB)
4p1r_validation.xml
PNG4p1r_multipercentile_validation.png.gz Display(165.99 KB)
4p1r_multipercentile_validation.png
SVG4p1r_multipercentile_validation.svg.gz Display(956.00 B)
4p1r_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4p1r_validation_2fo-fc_map_coef.cif.gz Display(670.84 KB)
4p1r_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4p1r_validation_fo-fc_map_coef.cif.gz Display(643.68 KB)
4p1r_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4p1r_validation_2fo-fc_map_coef.mtz Visualize(1.47 MB)
fo-fc (MTZ)4p1r_validation_fo-fc_map_coef.mtz Visualize(1.47 MB)

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PDB entries from 2024-07-24

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