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2GU8

Discovery of 2-Pyrimidyl-5-Amidothiophenes as Novel and Potent Inhibitors for AKT: Synthesis and SAR Studies

Resources
File formatFile name (file size)
PDBx/mmCIF2gu8.cif.gz Display(91.15 KB)
2gu8.cif
PDBx/mmJSONall2gu8.json.gz Display (Tree)(62.10 KB)
2gu8.json
no-atom2gu8-noatom.json.gz Display (Header)(13.95 KB)
2gu8-noatom.json
add only2gu8-plus.json.gz Display(3.52 KB)
2gu8-plus.json
PDBMLall2gu8.xml.gz Display(120.57 KB)
2gu8.xml
no-atom2gu8-noatom.xml.gz Display(27.33 KB)
2gu8-noatom.xml
ext-atom2gu8-extatom.xml.gz Display(69.63 KB)
2gu8-extatom.xml
pdb_nextgenallpdb_00002gu8_xyz-enrich.cif.gz Display(101.36 KB)
pdb_00002gu8_xyz-enrich.cif
no-atompdb_00002gu8_xyz-no-atom-enrich.xml.gz Display(38.63 KB)
pdb_00002gu8_xyz-no-atom-enrich.xml
ng-only2gu8-plus.json.gz Display(2.95 KB)
2gu8-plus.json
PDBpdb2gu8.ent.gz Display(67.20 KB)
pdb2gu8.ent
RDF2gu8.rdf.gz Visualize(82.22 KB)
2gu8.rdf
Structure factorsr2gu8sf.ent.gz Display(327.79 KB)
r2gu8sf.ent
Biological unit (mmCIF format)2gu8-assembly1.cif.gz Display(81.54 KB)
2gu8-assembly1.cif (A,C)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)2gu8.pdb1.gz Display(62.57 KB)
2gu8.pdb1 (A,C)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF2gu8_validation.pdf.gz Display(782.67 KB)
2gu8_validation.pdf
PDF-full2gu8_full_validation.pdf.gz Display(789.30 KB)
2gu8_full_validation.pdf
mmCIF2gu8_validation.cif.gz Display(26.97 KB)
2gu8_validation.cif
XML2gu8_validation.xml.gz Display(20.41 KB)
2gu8_validation.xml
PNG2gu8_multipercentile_validation.png.gz Display(166.35 KB)
2gu8_multipercentile_validation.png
SVG2gu8_multipercentile_validation.svg.gz Display(953.00 B)
2gu8_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)2gu8_validation_2fo-fc_map_coef.cif.gz Display(332.11 KB)
2gu8_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)2gu8_validation_fo-fc_map_coef.cif.gz Display(332.84 KB)
2gu8_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)2gu8_validation_2fo-fc_map_coef.mtz Visualize(538.13 KB)
fo-fc (MTZ)2gu8_validation_fo-fc_map_coef.mtz Visualize(538.13 KB)

238268

PDB entries from 2025-07-02

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