Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

9QFC

Tankyrase 2 ARC4 in complex with a pyrrolone-based inhibitor

This is a non-PDB format compatible entry.
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues64
DetailsRepeat: {"description":"ANK 10"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues64
DetailsRepeat: {"description":"ANK 11"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues64
DetailsRepeat: {"description":"ANK 12"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues16
DetailsRegion: {"description":"HIF1AN-binding","evidences":[{"source":"PubMed","id":"21251231","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues4
DetailsModified residue: {"description":"(3S)-3-hydroxyasparagine; by HIF1AN; partial","evidences":[{"source":"PubMed","id":"18936059","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues2
DetailsModified residue: {"description":"(3S)-3-hydroxyhistidine; by HIF1AN; partial","evidences":[{"source":"PubMed","id":"21251231","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

254227

PDB entries from 2026-05-27

PDB statisticsPDBj update infoContact PDBjnumon