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8TH3

Structure of AT118-H Nanobody Antagonist in Complex with the Angiotensin II Type I Receptor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0004945molecular_functionangiotensin type II receptor activity
A0005506molecular_functioniron ion binding
A0007186biological_processG protein-coupled receptor signaling pathway
A0009055molecular_functionelectron transfer activity
A0016020cellular_componentmembrane
A0019229biological_processregulation of vasoconstriction
A0020037molecular_functionheme binding
A0022900biological_processelectron transport chain
A0042597cellular_componentperiplasmic space
A0046872molecular_functionmetal ion binding
B0004930molecular_functionG protein-coupled receptor activity
B0004945molecular_functionangiotensin type II receptor activity
B0005506molecular_functioniron ion binding
B0007186biological_processG protein-coupled receptor signaling pathway
B0009055molecular_functionelectron transfer activity
B0016020cellular_componentmembrane
B0019229biological_processregulation of vasoconstriction
B0020037molecular_functionheme binding
B0022900biological_processelectron transport chain
B0042597cellular_componentperiplasmic space
B0046872molecular_functionmetal ion binding
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. ASVfLLTCLSIDRYLaI
ChainResidueDetails
AALA114-ILE130

site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. YACEVTH
ChainResidueDetails
DTYR194-HIS200
CTYR208-HIS214

site_idPS00324
Number of Residues9
DetailsASPARTOKINASE Aspartokinase signature. LlKYGGSSL
ChainResidueDetails
ALEU1316-LEU1324

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"description":"axial binding residue"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues29
DetailsTransmembrane: {"description":"Helical; Name=1","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues20
DetailsTopological domain: {"description":"Cytoplasmic","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues27
DetailsTransmembrane: {"description":"Helical; Name=2","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues32
DetailsTopological domain: {"description":"Extracellular","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues26
DetailsTransmembrane: {"description":"Helical; Name=3","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues23
DetailsTransmembrane: {"description":"Helical; Name=4","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues25
DetailsTransmembrane: {"description":"Helical; Name=5","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS2","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues28
DetailsTransmembrane: {"description":"Helical; Name=6","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI10
Number of Residues9
DetailsTopological domain: {"description":"Extracellular","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI11
Number of Residues25
DetailsTransmembrane: {"description":"Helical; Name=7","evidences":[{"source":"PubMed","id":"25913193","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"26420482","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4YAY","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4ZUD","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI12
Number of Residues5
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000305"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000305"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI13
Number of Residues1
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"source":"PubMed","id":"30639100","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"32079768","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"6DO1","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"6OS0","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI14
Number of Residues1
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

239149

PDB entries from 2025-07-23

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