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8RIY

Human NUDT5 with ibrutinib derivative

This is a non-PDB format compatible entry.
Functional Information from PROSITE/UniProt
site_idPS00893
Number of Residues22
DetailsNUDIX_BOX Nudix box signature. GliddgEtpeaAAlRELeEEtG
ChainResidueDetails
AAAGLY97-GLY118

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: in other chain => ECO:0000269|PubMed:17052728, ECO:0000269|PubMed:18462755, ECO:0000269|PubMed:21768126
ChainResidueDetails
AAATRP28
AAAARG84
BBBTRP28
BBBARG84

site_idSWS_FT_FI2
Number of Residues12
DetailsBINDING: BINDING => ECO:0000269|PubMed:17052728, ECO:0000269|PubMed:18462755, ECO:0000269|PubMed:21768126
ChainResidueDetails
AAATRP46
BBBGLU112
BBBGLU116
BBBGLU166
AAAARG51
AAAALA96
AAAGLU112
AAAGLU116
AAAGLU166
BBBTRP46
BBBARG51
BBBALA96

site_idSWS_FT_FI3
Number of Residues4
DetailsBINDING: in other chain => ECO:0000269|PubMed:17052728
ChainResidueDetails
AAALEU98
AAAASP133
BBBLEU98
BBBASP133

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: N-acetylmethionine => ECO:0007744|PubMed:19413330, ECO:0007744|PubMed:20068231, ECO:0007744|PubMed:21406692, ECO:0007744|PubMed:22223895
ChainResidueDetails
AAAMET1
BBBMET1

site_idSWS_FT_FI5
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:21406692, ECO:0007744|PubMed:23186163
ChainResidueDetails
AAASER3
BBBSER3

site_idSWS_FT_FI6
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:20068231
ChainResidueDetails
AAASER10
BBBSER10

site_idSWS_FT_FI7
Number of Residues2
DetailsMOD_RES: Phosphothreonine => ECO:0000269|PubMed:27257257
ChainResidueDetails
AAATHR45
BBBTHR45

site_idSWS_FT_FI8
Number of Residues2
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:15592455
ChainResidueDetails
AAATYR74
BBBTYR74

site_idSWS_FT_FI9
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
AAALYS42
BBBLYS42

221716

PDB entries from 2024-06-26

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