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7W7O

The crystal structure of human Calpain-1 protease core in complex with 14a

Functional Information from GO Data
ChainGOidnamespacecontents
A0004198molecular_functioncalcium-dependent cysteine-type endopeptidase activity
A0006508biological_processproteolysis
Functional Information from PROSITE/UniProt
site_idPS00139
Number of Residues12
DetailsTHIOL_PROTEASE_CYS Eukaryotic thiol (cysteine) proteases cysteine active site. QGaLGDCWLlAA
ChainResidueDetails
AGLN109-ALA120

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: ACT_SITE => ECO:0000250
ChainResidueDetails
ACYS115
AHIS272
AASN296

site_idSWS_FT_FI2
Number of Residues5
DetailsBINDING: BINDING => ECO:0000305
ChainResidueDetails
AGLN109
AASP114
AASN316
AASP318
AASP323

site_idSWS_FT_FI3
Number of Residues1
DetailsSITE: Cleavage; for 75 kDa form
ChainResidueDetails
AGLY27

site_idSWS_FT_FI4
Number of Residues1
DetailsMOD_RES: Phosphothreonine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATHR354

223532

PDB entries from 2024-08-07

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