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7PDT

Crystal structure of a mutated form of RXRalpha ligand binding domain in complex with BMS649 and a coactivator fragment

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003707molecular_functionnuclear steroid receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
B0003677molecular_functionDNA binding
B0003707molecular_functionnuclear steroid receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
B0008270molecular_functionzinc ion binding
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues40
DetailsRegion: {"description":"Required for nuclear export","evidences":[{"source":"UniProtKB","id":"P19793","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P19793","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 2"}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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