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7LB3

Crystal structure of the second bromodomain (BD2) of human TAF1 bound to ZS1-580

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue XXS A 1701
ChainResidue
ATRP1526
ATYR1601
ATHR1605
AEDO1702
AHOH1824
AHOH1825
AHOH1894
APRO1527
AHIS1530
APRO1531
AVAL1532
AASN1533
APHE1536
AASN1583
ATYR1589

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 1702
ChainResidue
AARG1565
AASP1608
AXXS1701
AHOH1802
AHOH1806
AHOH1822

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFhhpvNkkfvp..DYYkvIvnpMdletIrkniskhk..Yqsresflddvnl.IlaNSvkY
ChainResidueDetails
ASER1525-TYR1582

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PDB entries from 2024-10-09

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