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7L73

Crystal structure of the first bromodomain (BD1) of human BRDT bound to ERK5-IN-1

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue VYJ A 201
ChainResidue
ATRP50
AGLN120
AHOH315
AHOH322
AHOH355
AHOH392
APRO51
ALYS60
ALEU61
ALEU63
ASER103
ATYR106
AASN109
APRO111

site_idAC2
Number of Residues14
Detailsbinding site for residue VYJ A 202
ChainResidue
ALYS41
ATRP44
ALYS45
AGLN62
ALEU63
AASP65
AILE95
AASN99
ATYR108
AMET127
ALEU130
ASER131
AMET133
AHOH310

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFqrpvDavklqlpDYYtiIknpMdlntIkkrlenky..Yakaseciedfnt.MfsNCylY
ChainResidueDetails
ASER49-TYR108

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsBINDING: BINDING => ECO:0000269|PubMed:22901802, ECO:0007744|PDB:4FLP
ChainResidueDetails
AGLU96

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Histone H4K5ac binding => ECO:0000250|UniProtKB:Q91Y44
ChainResidueDetails
AGLU96
AMET101

221716

PDB entries from 2024-06-26

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