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7L73

Crystal structure of the first bromodomain (BD1) of human BRDT bound to ERK5-IN-1

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue VYJ A 201
ChainResidue
ATRP50
AGLN120
AHOH315
AHOH322
AHOH355
AHOH392
APRO51
ALYS60
ALEU61
ALEU63
ASER103
ATYR106
AASN109
APRO111

site_idAC2
Number of Residues14
Detailsbinding site for residue VYJ A 202
ChainResidue
ALYS41
ATRP44
ALYS45
AGLN62
ALEU63
AASP65
AILE95
AASN99
ATYR108
AMET127
ALEU130
ASER131
AMET133
AHOH310

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFqrpvDavklqlpDYYtiIknpMdlntIkkrlenky..Yakaseciedfnt.MfsNCylY
ChainResidueDetails
ASER49-TYR108

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"22901802","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4FLP","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsSite: {"description":"Histone H4K5ac binding","evidences":[{"source":"UniProtKB","id":"Q91Y44","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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