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7EVJ

Crystal structure of CBP bromodomain liganded with 9c

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue JE9 A 1201
ChainResidue
ALEU1109
AHOH1302
AHOH1322
APRO1110
AGLN1113
ALEU1120
AILE1122
AASN1168
AARG1173
AVAL1174
APO41202

site_idAC2
Number of Residues5
Detailsbinding site for residue PO4 A 1202
ChainResidue
ASER1172
AARG1173
AARG1173
AJE91201
AHOH1326

site_idAC3
Number of Residues3
Detailsbinding site for residue GOL A 1203
ChainResidue
AGLN1146
ATRP1158
AASN1162

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-07-10

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