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7ENZ

Crystal structure of Phenanthredinone moiety in complex with the second bromodomain of BRD2 (BRD2-BD2).

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue LDR A 701
ChainResidue
APRO371
AVAL376
AASN429
AHOH805

site_idAC2
Number of Residues7
Detailsbinding site for residue PGE A 702
ChainResidue
AHOH862
AHOH886
APRO347
ALEU350
ALYS351
AMET403
AHOH821

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues109
DetailsDomain: {"description":"Bromo 2","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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