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7DXG

Structure of SAR7334-bound TRPC6 at 2.9 angstrom

Functional Information from GO Data
ChainGOidnamespacecontents
A0003779molecular_functionactin binding
A0005216molecular_functionmonoatomic ion channel activity
A0005261molecular_functionmonoatomic cation channel activity
A0005262molecular_functioncalcium channel activity
A0005515molecular_functionprotein binding
A0005737cellular_componentcytoplasm
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0006812biological_processmonoatomic cation transport
A0006816biological_processcalcium ion transport
A0007204biological_processpositive regulation of cytosolic calcium ion concentration
A0007338biological_processsingle fertilization
A0015279molecular_functionstore-operated calcium channel activity
A0016020cellular_componentmembrane
A0030182biological_processneuron differentiation
A0030276molecular_functionclathrin binding
A0032414biological_processpositive regulation of ion transmembrane transporter activity
A0034220biological_processmonoatomic ion transmembrane transport
A0034703cellular_componentcation channel complex
A0036057cellular_componentslit diaphragm
A0042803molecular_functionprotein homodimerization activity
A0042805molecular_functionactinin binding
A0045666biological_processpositive regulation of neuron differentiation
A0050774biological_processnegative regulation of dendrite morphogenesis
A0051117molecular_functionATPase binding
A0051480biological_processregulation of cytosolic calcium ion concentration
A0051928biological_processpositive regulation of calcium ion transport
A0055085biological_processtransmembrane transport
A0070301biological_processcellular response to hydrogen peroxide
A0070588biological_processcalcium ion transmembrane transport
A0070679molecular_functioninositol 1,4,5 trisphosphate binding
A0071456biological_processcellular response to hypoxia
B0003779molecular_functionactin binding
B0005216molecular_functionmonoatomic ion channel activity
B0005261molecular_functionmonoatomic cation channel activity
B0005262molecular_functioncalcium channel activity
B0005515molecular_functionprotein binding
B0005737cellular_componentcytoplasm
B0005886cellular_componentplasma membrane
B0006811biological_processmonoatomic ion transport
B0006812biological_processmonoatomic cation transport
B0006816biological_processcalcium ion transport
B0007204biological_processpositive regulation of cytosolic calcium ion concentration
B0007338biological_processsingle fertilization
B0015279molecular_functionstore-operated calcium channel activity
B0016020cellular_componentmembrane
B0030182biological_processneuron differentiation
B0030276molecular_functionclathrin binding
B0032414biological_processpositive regulation of ion transmembrane transporter activity
B0034220biological_processmonoatomic ion transmembrane transport
B0034703cellular_componentcation channel complex
B0036057cellular_componentslit diaphragm
B0042803molecular_functionprotein homodimerization activity
B0042805molecular_functionactinin binding
B0045666biological_processpositive regulation of neuron differentiation
B0050774biological_processnegative regulation of dendrite morphogenesis
B0051117molecular_functionATPase binding
B0051480biological_processregulation of cytosolic calcium ion concentration
B0051928biological_processpositive regulation of calcium ion transport
B0055085biological_processtransmembrane transport
B0070301biological_processcellular response to hydrogen peroxide
B0070588biological_processcalcium ion transmembrane transport
B0070679molecular_functioninositol 1,4,5 trisphosphate binding
B0071456biological_processcellular response to hypoxia
C0003779molecular_functionactin binding
C0005216molecular_functionmonoatomic ion channel activity
C0005261molecular_functionmonoatomic cation channel activity
C0005262molecular_functioncalcium channel activity
C0005515molecular_functionprotein binding
C0005737cellular_componentcytoplasm
C0005886cellular_componentplasma membrane
C0006811biological_processmonoatomic ion transport
C0006812biological_processmonoatomic cation transport
C0006816biological_processcalcium ion transport
C0007204biological_processpositive regulation of cytosolic calcium ion concentration
C0007338biological_processsingle fertilization
C0015279molecular_functionstore-operated calcium channel activity
C0016020cellular_componentmembrane
C0030182biological_processneuron differentiation
C0030276molecular_functionclathrin binding
C0032414biological_processpositive regulation of ion transmembrane transporter activity
C0034220biological_processmonoatomic ion transmembrane transport
C0034703cellular_componentcation channel complex
C0036057cellular_componentslit diaphragm
C0042803molecular_functionprotein homodimerization activity
C0042805molecular_functionactinin binding
C0045666biological_processpositive regulation of neuron differentiation
C0050774biological_processnegative regulation of dendrite morphogenesis
C0051117molecular_functionATPase binding
C0051480biological_processregulation of cytosolic calcium ion concentration
C0051928biological_processpositive regulation of calcium ion transport
C0055085biological_processtransmembrane transport
C0070301biological_processcellular response to hydrogen peroxide
C0070588biological_processcalcium ion transmembrane transport
C0070679molecular_functioninositol 1,4,5 trisphosphate binding
C0071456biological_processcellular response to hypoxia
D0003779molecular_functionactin binding
D0005216molecular_functionmonoatomic ion channel activity
D0005261molecular_functionmonoatomic cation channel activity
D0005262molecular_functioncalcium channel activity
D0005515molecular_functionprotein binding
D0005737cellular_componentcytoplasm
D0005886cellular_componentplasma membrane
D0006811biological_processmonoatomic ion transport
D0006812biological_processmonoatomic cation transport
D0006816biological_processcalcium ion transport
D0007204biological_processpositive regulation of cytosolic calcium ion concentration
D0007338biological_processsingle fertilization
D0015279molecular_functionstore-operated calcium channel activity
D0016020cellular_componentmembrane
D0030182biological_processneuron differentiation
D0030276molecular_functionclathrin binding
D0032414biological_processpositive regulation of ion transmembrane transporter activity
D0034220biological_processmonoatomic ion transmembrane transport
D0034703cellular_componentcation channel complex
D0036057cellular_componentslit diaphragm
D0042803molecular_functionprotein homodimerization activity
D0042805molecular_functionactinin binding
D0045666biological_processpositive regulation of neuron differentiation
D0050774biological_processnegative regulation of dendrite morphogenesis
D0051117molecular_functionATPase binding
D0051480biological_processregulation of cytosolic calcium ion concentration
D0051928biological_processpositive regulation of calcium ion transport
D0055085biological_processtransmembrane transport
D0070301biological_processcellular response to hydrogen peroxide
D0070588biological_processcalcium ion transmembrane transport
D0070679molecular_functioninositol 1,4,5 trisphosphate binding
D0071456biological_processcellular response to hypoxia
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues480
DetailsTransmembrane: {"description":"Helical","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues136
DetailsTopological domain: {"description":"Cytoplasmic","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues192
DetailsTopological domain: {"description":"Extracellular","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues116
DetailsRepeat: {"description":"ANK 1"}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues116
DetailsRepeat: {"description":"ANK 2"}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues104
DetailsRepeat: {"description":"ANK 3"}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues116
DetailsRepeat: {"description":"ANK 4"}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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