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7DN4

The crystal structure of Cpd8 in complex with BPTF bromodomain

Functional Information from GO Data
ChainGOidnamespacecontents
A0006357biological_processregulation of transcription by RNA polymerase II
A0016589cellular_componentNURF complex
B0006357biological_processregulation of transcription by RNA polymerase II
B0016589cellular_componentNURF complex
C0006357biological_processregulation of transcription by RNA polymerase II
C0016589cellular_componentNURF complex
D0006357biological_processregulation of transcription by RNA polymerase II
D0016589cellular_componentNURF complex
E0006357biological_processregulation of transcription by RNA polymerase II
E0016589cellular_componentNURF complex
F0006357biological_processregulation of transcription by RNA polymerase II
F0016589cellular_componentNURF complex
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue JC3 A 3001
ChainResidue
ATRP2824
APRO2825
APHE2826
APRO2829
AALA2835
ATYR2880
AASN2881
EMET2796

site_idAC2
Number of Residues8
Detailsbinding site for residue JC3 B 3001
ChainResidue
BPRO2825
BPHE2826
BPRO2829
BALA2835
BCYS2877
BTYR2880
BASN2881
BTRP2824

site_idAC3
Number of Residues9
Detailsbinding site for residue JC3 C 3001
ChainResidue
CTRP2824
CPRO2825
CPHE2826
CPRO2829
CVAL2830
CALA2835
CTYR2880
CASN2881
CPHE2887

site_idAC4
Number of Residues8
Detailsbinding site for residue JC3 D 3001
ChainResidue
DTRP2824
DPRO2825
DPRO2829
DALA2835
DCYS2877
DTYR2880
DASN2881
DPHE2887

site_idAC5
Number of Residues9
Detailsbinding site for residue JC3 E 3001
ChainResidue
ETRP2824
EPRO2825
EPHE2826
EPRO2829
EVAL2830
EALA2835
ETYR2880
EASN2881
EPHE2887

site_idAC6
Number of Residues7
Detailsbinding site for residue JC3 F 3001
ChainResidue
FTRP2824
FPRO2825
FPHE2826
FPRO2829
FALA2835
FTYR2880
FASN2881

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFlepvDpndap..DYYgvIkepMdlatMeervqrry..Yekltefvadmtk.IfdNCryY
ChainResidueDetails
AALA2823-TYR2880

222415

PDB entries from 2024-07-10

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