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7CLZ

Crystal structure of Alp1U W187F/Y247F in complex with fluostatin C

Functional Information from GO Data
ChainGOidnamespacecontents
A0003824molecular_functioncatalytic activity
B0003824molecular_functioncatalytic activity
C0003824molecular_functioncatalytic activity
D0003824molecular_functioncatalytic activity
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue DY9 A 401
ChainResidue
ATRP72
AHIS300
ATYR301
AHOH503
AASP137
AMET141
ATHR162
ATRP186
APHE187
ALEU211
AASN214
AVAL299

site_idAC2
Number of Residues3
Detailsbinding site for residue NA A 402
ChainResidue
AARG33
AARG37
ASER45

site_idAC3
Number of Residues10
Detailsbinding site for residue MLT A 403
ChainResidue
AHIS201
AGLY202
AASN235
APRO237
AHOH519
AHOH569
DARG205
DGLN219
DVAL222
DARG227

site_idAC4
Number of Residues4
Detailsbinding site for residue NA B 401
ChainResidue
BARG33
BARG37
BARG44
BSER45

site_idAC5
Number of Residues9
Detailsbinding site for residue MLT B 402
ChainResidue
BHIS201
BGLY202
BASN235
BSER236
BPRO237
BHOH501
CARG205
CGLN219
CARG227

site_idAC6
Number of Residues9
Detailsbinding site for residue MLT B 403
ChainResidue
BLYS105
BPRO106
BALA107
BTYR110
BGLN238
BARG241
BALA242
BARG245
BHOH577

site_idAC7
Number of Residues12
Detailsbinding site for residue DY9 C 401
ChainResidue
CTRP72
CASP137
CTHR162
CTRP186
CPHE187
CLEU211
CASN214
CPHE247
CVAL299
CHIS300
CTYR301
CHOH505

site_idAC8
Number of Residues5
Detailsbinding site for residue BO3 C 402
ChainResidue
CLYS105
CPRO106
CALA107
CARG241
CARG245

site_idAC9
Number of Residues11
Detailsbinding site for residue DY9 D 401
ChainResidue
DTRP72
DASP137
DTHR162
DTRP186
DPHE187
DLEU211
DASN214
DPHE247
DHIS300
DTYR301
DHOH502

site_idAD1
Number of Residues4
Detailsbinding site for residue BO3 D 402
ChainResidue
DPRO106
DALA107
DARG241
DARG245

site_idAD2
Number of Residues11
Detailsbinding site for residue MLT D 403
ChainResidue
BHOH532
CGLY202
CHIS206
CHOH539
CHOH555
DGLY202
DARG205
DHIS206
DHOH509
DHOH533
DHOH556

223532

PDB entries from 2024-08-07

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