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7C60

Crystal structure of Keap1 in complex with monoethyl fumarate (MEF)

Functional Information from GO Data
ChainGOidnamespacecontents
A0008134molecular_functiontranscription factor binding
A0016567biological_processprotein ubiquitination
A0031463cellular_componentCul3-RING ubiquitin ligase complex
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue NF3 A 801
ChainResidue
AVAL369
AVAL370
AGLY371
AGLY372
AHOH1063
AHOH1089

site_idAC2
Number of Residues5
Detailsbinding site for residue ACT A 802
ChainResidue
AHOH996
AHOH1027
AARG380
AASN382
AASN414

site_idAC3
Number of Residues5
Detailsbinding site for residue NF3 A 803
ChainResidue
ATYR525
AGLN530
ASER555
ATYR572
AHOH1000

site_idAC4
Number of Residues10
Detailsbinding site for residue SO4 A 804
ChainResidue
AILE435
AHIS437
ASER438
ASER439
AARG494
AHOH904
AHOH917
AHOH966
AHOH1017
AHOH1066

site_idAC5
Number of Residues7
Detailsbinding site for residue SO4 A 805
ChainResidue
ACYS434
AHIS436
AARG459
AARG494
AARG498
AHOH963
AHOH975

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues45
DetailsRepeat: {"description":"Kelch 1"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues50
DetailsRepeat: {"description":"Kelch 2"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues46
DetailsRepeat: {"description":"Kelch 3"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues46
DetailsRepeat: {"description":"Kelch 4"}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues45
DetailsRepeat: {"description":"Kelch 5"}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues46
DetailsRepeat: {"description":"Kelch 6"}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues1
DetailsSite: {"description":"Sensor for electrophilic agents","evidences":[{"source":"PubMed","id":"20498371","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues2
DetailsModified residue: {"description":"S-(2-succinyl)cysteine","evidences":[{"source":"PubMed","id":"22014577","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues1
DetailsModified residue: {"description":"S-cGMP-cysteine","evidences":[{"source":"PubMed","id":"20498371","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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