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6ZBZ

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

Functional Information from GO Data
ChainGOidnamespacecontents
A0016055biological_processWnt signaling pathway
B0016055biological_processWnt signaling pathway
C0016055biological_processWnt signaling pathway
D0016055biological_processWnt signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue QE5 A 401
ChainResidue
APHE259
CGLN301
CHOH599
ALEU260
AGLY261
AILE262
AARG320
AVAL323
AHIS324
AHOH533
CLEU300

site_idAC2
Number of Residues12
Detailsbinding site for residue QE5 B 401
ChainResidue
BPHE259
BLEU260
BGLY261
BILE262
BLEU319
BARG320
BVAL323
BHIS324
BHOH529
CASN253
CGLU255
CPRO328

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO B 402
ChainResidue
BGLN267
BSER268
BASN269
BMET310
BSER311
BHOH522

site_idAC4
Number of Residues13
Detailsbinding site for residue QE5 C 401
ChainResidue
BMET310
BASP314
BVAL318
BGLU321
CPHE259
CLEU260
CGLY261
CILE262
CVAL316
CLEU319
CARG320
CVAL323
CHIS324

site_idAC5
Number of Residues6
Detailsbinding site for residue EDO C 402
ChainResidue
CILE322
CLYS325
CPRO326
CHOH507
CHOH532
CHOH556

site_idAC6
Number of Residues2
Detailsbinding site for residue EDO C 403
ChainResidue
AASN269
AASP273

site_idAC7
Number of Residues11
Detailsbinding site for residue QE5 D 401
ChainResidue
AASN303
AGLU304
AILE305
DLEU260
DGLY261
DILE262
DLEU319
DARG320
DVAL323
DHIS324
DHOH520

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Symmetric dimethylarginine; by PRMT7; alternate","evidences":[{"source":"PubMed","id":"23150776","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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