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6YTM

Human Brd2(BD2) L383V mutant in complex with ET-JQ1-OMe

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue PMW A 501
ChainResidue
APRO371
ATYR428
AASN429
AHIS433
AVAL435
AHOH614
BSER379

site_idAC2
Number of Residues3
Detailsbinding site for residue PXN A 502
ChainResidue
AHOH647
AASP407
ALYS441

site_idAC3
Number of Residues4
Detailsbinding site for residue PXN A 503
ChainResidue
APRO431
AALA437
AHOH678
BASP444

site_idAC4
Number of Residues9
Detailsbinding site for residue PMW B 501
ChainResidue
BPRO371
BPHE372
BVAL376
BTYR428
BASN429
BHIS433
BASP434
BVAL435
BHOH611

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalgvhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

249697

PDB entries from 2026-02-25

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