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6X0P

Ash1L SET domain Q2265A mutant in complex with AS-5

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0042054molecular_functionhistone methyltransferase activity
B0005634cellular_componentnucleus
B0042054molecular_functionhistone methyltransferase activity
C0005634cellular_componentnucleus
C0042054molecular_functionhistone methyltransferase activity
D0005634cellular_componentnucleus
D0042054molecular_functionhistone methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue UK7 A 2301
ChainResidue
AHIS2193
AILE2279
AGLY2280
AGLY2281
AHOH2464
AHOH2562
AHOH2566
ACYS2195
ATYR2255
AASN2256
ASER2259
APHE2260
AASN2261
ALYS2264
AGLN2266

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 2302
ChainResidue
ACYS2091
ACYS2093
ACYS2104
ACYS2108

site_idAC3
Number of Residues4
Detailsbinding site for residue ZN A 2303
ChainResidue
ACYS2104
ACYS2117
ACYS2122
ACYS2128

site_idAC4
Number of Residues4
Detailsbinding site for residue ZN A 2304
ChainResidue
ACYS2220
ACYS2268
ACYS2270
ACYS2275

site_idAC5
Number of Residues23
Detailsbinding site for residue SAM A 2305
ChainResidue
ALYS2150
AGLY2151
ATRP2152
ASER2191
AASP2192
AHIS2193
ATYR2194
AARG2214
APHE2215
AASN2217
AHIS2218
ATYR2255
AGLN2266
ALEU2267
ACYS2268
ALYS2269
AILE2279
AHOH2413
AHOH2436
AHOH2450
AHOH2472
AHOH2482
AHOH2570

site_idAC6
Number of Residues14
Detailsbinding site for residue UK7 B 2301
ChainResidue
BHIS2193
BCYS2195
BTYR2255
BASN2256
BSER2259
BPHE2260
BASN2261
BVAL2262
BLYS2264
BGLN2266
BILE2278
BILE2279
BGLY2280
BSAM2305

site_idAC7
Number of Residues4
Detailsbinding site for residue ZN B 2302
ChainResidue
BCYS2091
BCYS2093
BCYS2104
BCYS2108

site_idAC8
Number of Residues4
Detailsbinding site for residue ZN B 2303
ChainResidue
BCYS2104
BCYS2117
BCYS2122
BCYS2128

site_idAC9
Number of Residues4
Detailsbinding site for residue ZN B 2304
ChainResidue
BCYS2220
BCYS2268
BCYS2270
BCYS2275

site_idAD1
Number of Residues22
Detailsbinding site for residue SAM B 2305
ChainResidue
BLYS2150
BGLY2151
BTRP2152
BSER2191
BASP2192
BHIS2193
BTYR2194
BARG2214
BPHE2215
BASN2217
BHIS2218
BTYR2255
BGLN2266
BLEU2267
BCYS2268
BLYS2269
BILE2279
BUK72301
BHOH2413
BHOH2424
BHOH2430
BHOH2501

site_idAD2
Number of Residues15
Detailsbinding site for residue UK7 C 2301
ChainResidue
CCYS2195
CTYR2255
CASN2256
CSER2259
CPHE2260
CASN2261
CLYS2264
CGLN2266
CILE2278
CILE2279
CGLY2280
CHOH2456
CHOH2480
CHOH2501
CHIS2193

site_idAD3
Number of Residues4
Detailsbinding site for residue ZN C 2302
ChainResidue
CCYS2091
CCYS2093
CCYS2104
CCYS2108

site_idAD4
Number of Residues4
Detailsbinding site for residue ZN C 2303
ChainResidue
CCYS2104
CCYS2117
CCYS2122
CCYS2128

site_idAD5
Number of Residues4
Detailsbinding site for residue ZN C 2304
ChainResidue
CCYS2220
CCYS2268
CCYS2270
CCYS2275

site_idAD6
Number of Residues23
Detailsbinding site for residue SAM C 2305
ChainResidue
CLYS2150
CGLY2151
CTRP2152
CSER2191
CASP2192
CHIS2193
CTYR2194
CARG2214
CPHE2215
CASN2217
CHIS2218
CTYR2255
CGLN2266
CLEU2267
CCYS2268
CLYS2269
CILE2279
CHOH2414
CHOH2436
CHOH2477
CHOH2483
CHOH2542
CHOH2583

site_idAD7
Number of Residues16
Detailsbinding site for residue UK7 D 2301
ChainResidue
DHIS2193
DCYS2195
DTYR2255
DASN2256
DSER2259
DPHE2260
DASN2261
DVAL2262
DLYS2264
DGLN2266
DILE2278
DILE2279
DGLY2280
DGLY2281
DSAM2305
DHOH2562

site_idAD8
Number of Residues4
Detailsbinding site for residue ZN D 2302
ChainResidue
DCYS2091
DCYS2093
DCYS2104
DCYS2108

site_idAD9
Number of Residues4
Detailsbinding site for residue ZN D 2303
ChainResidue
DCYS2104
DCYS2117
DCYS2122
DCYS2128

site_idAE1
Number of Residues4
Detailsbinding site for residue ZN D 2304
ChainResidue
DCYS2220
DCYS2268
DCYS2270
DCYS2275

site_idAE2
Number of Residues22
Detailsbinding site for residue SAM D 2305
ChainResidue
DLYS2150
DTRP2152
DSER2191
DASP2192
DHIS2193
DTYR2194
DARG2214
DPHE2215
DASN2217
DHIS2218
DTYR2255
DGLN2266
DLEU2267
DCYS2268
DLYS2269
DILE2279
DUK72301
DHOH2421
DHOH2459
DHOH2484
DHOH2528
DHOH2576

222415

PDB entries from 2024-07-10

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