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6VLM

Core Catalytic Domain of HIV Integrase in complex with virtual screening hit

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue R2D A 301
ChainResidue
AGLN168
AALA169
AGLU170
AHIS171
ATHR174
ATHR210
BALA128
BTRP132
BR2D302

site_idAC2
Number of Residues7
Detailsbinding site for residue R2D B 301
ChainResidue
ATHR125
AALA128
ATRP132
BALA169
BGLU170
BHIS171
BTHR174

site_idAC3
Number of Residues6
Detailsbinding site for residue R2D B 302
ChainResidue
AR2D301
BLYS127
BALA128
BTRP131
BTRP132
BHOH412

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP64
AASP116
BASP64
BASP116

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152
BGLU152

221371

PDB entries from 2024-06-19

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