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6VLM

Core Catalytic Domain of HIV Integrase in complex with virtual screening hit

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue R2D A 301
ChainResidue
AGLN168
AALA169
AGLU170
AHIS171
ATHR174
ATHR210
BALA128
BTRP132
BR2D302

site_idAC2
Number of Residues7
Detailsbinding site for residue R2D B 301
ChainResidue
ATHR125
AALA128
ATRP132
BALA169
BGLU170
BHIS171
BTHR174

site_idAC3
Number of Residues6
Detailsbinding site for residue R2D B 302
ChainResidue
AR2D301
BLYS127
BALA128
BTRP131
BTRP132
BHOH412

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBinding site: {"evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P04585","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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