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6VJD

Estrogen Receptor Alpha Ligand Binding Domain in Complex with Lasofoxifene

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue C3D A 601
ChainResidue
AMET343
ALEU525
AASN532
AVAL533
AHOH729
ALEU346
AALA350
AASP351
AGLU353
ATRP383
ALEU387
AARG394
AHIS524

site_idAC2
Number of Residues13
Detailsbinding site for residue C3D B 601
ChainResidue
BMET343
BLEU346
BTHR347
BALA350
BASP351
BGLU353
BLEU387
BARG394
BHIS524
BLEU525
BASN532
BVAL533
BHOH745

site_idAC3
Number of Residues12
Detailsbinding site for residue C3D C 601
ChainResidue
CLEU346
CTHR347
CALA350
CASP351
CGLU353
CTRP383
CLEU387
CARG394
CLEU525
CASN532
CVAL533
CHOH773

site_idAC4
Number of Residues14
Detailsbinding site for residue C3D D 601
ChainResidue
DMET343
DLEU346
DTHR347
DALA350
DASP351
DGLU353
DTRP383
DLEU387
DARG394
DHIS524
DLEU525
DASN532
DVAL533
DHOH723

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537
BTYR537
CTYR537
DTYR537

site_idSWS_FT_FI2
Number of Residues4
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447
CCYS447
DCYS447

219869

PDB entries from 2024-05-15

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