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6V16

Crystal structure of the bromodomain of human BRD7 bound to TP472

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue QMG A 301
ChainResidue
APHE155
APHE158
AILE164
AASN211
ATYR217
AHOH411
AHOH419
AHOH451
AHOH453

site_idAC2
Number of Residues2
Detailsbinding site for residue EDO A 302
ChainResidue
ALYS197
ALYS201

site_idAC3
Number of Residues11
Detailsbinding site for residue QMG B 301
ChainResidue
AARG236
ASER239
AHOH427
AHOH441
BPHE155
BPHE156
BVAL160
BILE164
BASN211
BTYR217
BHOH402

site_idAC4
Number of Residues2
Detailsbinding site for residue HEZ B 302
ChainResidue
BMET170
BILE171

site_idAC5
Number of Residues2
Detailsbinding site for residue GOL B 303
ChainResidue
BLYS197
BLYS201

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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