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6UOC

Crystal structure of Danio rerio histone deacetylase 6 catalytic domain 1 (CD1) K330L mutant complexed with Givinostat

Functional Information from GO Data
ChainGOidnamespacecontents
A0000118cellular_componenthistone deacetylase complex
A0004407molecular_functionhistone deacetylase activity
A0006325biological_processchromatin organization
A0016575biological_processhistone deacetylation
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 601
ChainResidue
AHIS345
ALYS348
ASER378
AGLY381
AASP382
AHOH940

site_idAC2
Number of Residues2
Detailsbinding site for residue EDO A 602
ChainResidue
ASER150
AHOH733

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 603
ChainResidue
AGLY327
AGLY332
AMET333
AGLN334
AHOH709
AILE326

site_idAC4
Number of Residues4
Detailsbinding site for residue ZN A 604
ChainResidue
AASP230
AHIS232
AASP323
AQCM607

site_idAC5
Number of Residues5
Detailsbinding site for residue K A 605
ChainResidue
AASP228
AASP230
AHIS232
ASER251
AVAL252

site_idAC6
Number of Residues6
Detailsbinding site for residue K A 606
ChainResidue
APHE241
AASP244
AVAL247
ATYR280
AHOH825
AHOH829

site_idAC7
Number of Residues14
Detailsbinding site for residue QCM A 607
ChainResidue
AGLU94
AGLU97
ASER150
AHIS192
AHIS193
APHE202
AASP230
AHIS232
ATRP261
AASP323
ALEU330
ATYR363
AZN604
AHOH828

223166

PDB entries from 2024-07-31

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