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6U6F

The crystal structure of anti-apoptotic Mcl-1 protein in complex with 2, 5-substituted benzoic acid inhibitor 21

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
C0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue PZY A 401
ChainResidue
AMET231
ALEU246
AMET250
AARG263
ATHR266
ALEU267
CGLY230
CARG233
CPZY401

site_idAC2
Number of Residues3
Detailsbinding site for residue PZY A 402
ChainResidue
AHIS252
CLYS234
CPZY401

site_idAC3
Number of Residues12
Detailsbinding site for residue PZY B 401
ChainResidue
BALA227
BGLY230
BMET231
BMET231
BLEU246
BSER247
BMET250
BVAL253
BARG263
BTHR266
BPHE270
BLEU290

site_idAC4
Number of Residues10
Detailsbinding site for residue PZY C 401
ChainResidue
AGLY230
AMET231
AARG233
APZY401
APZY402
CMET231
CVAL253
CPHE254
CARG263
CTHR266

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues9
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS194
ALYS197
BLYS194
BLYS197
CLYS194
CLYS197

218853

PDB entries from 2024-04-24

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