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6TLQ

ROR(gamma)t ligand binding domain in complex with cholesterol and allosteric ligand Glenmark

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue CLR A 601
ChainResidue
AGLN286
ACYS320
AHIS323
AMET365
ALEU391
ALEU396
APHE486
AGOL603
AHOH778

site_idAC2
Number of Residues17
Detailsbinding site for residue MJE A 602
ChainResidue
ATRP317
ALEU324
ATHR325
AILE328
AGLN329
ALEU353
ALYS354
AMET358
ALEU483
AGLN484
AGLN495
AALA496
AALA497
APHE498
ATYR502
ALEU505
APHE506

site_idAC3
Number of Residues6
Detailsbinding site for residue GOL A 603
ChainResidue
APHE377
APHE378
AGLU379
ACLR601
AHOH708
AHOH730

site_idAC4
Number of Residues3
Detailsbinding site for residue GOL A 604
ChainResidue
ACYS345
AGLN346
AHOH706

site_idAC5
Number of Residues6
Detailsbinding site for residue GOL A 605
ChainResidue
AARG296
ATHR306
AARG310
AHIS411
AHOH703
AHOH759

218853

PDB entries from 2024-04-24

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