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6THV

X-ray structure of the Danio rerio histone deacetylase 6 (HDAC6; catalytic domain 2) in complex with Tubastatin A

Functional Information from GO Data
ChainGOidnamespacecontents
A0000118cellular_componenthistone deacetylase complex
A0004407molecular_functionhistone deacetylase activity
A0006325biological_processchromatin organization
A0016575biological_processhistone deacetylation
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue ZN A 801
ChainResidue
AASP612
AHIS614
AASP705
AN9W813
AHOH903

site_idAC2
Number of Residues5
Detailsbinding site for residue K A 802
ChainResidue
ALEU634
AASP610
AASP612
AHIS614
ASER633

site_idAC3
Number of Residues6
Detailsbinding site for residue K A 803
ChainResidue
APHE623
AASP626
AVAL629
ATYR662
AHOH985
AHOH1030

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 804
ChainResidue
AHIS684
ALEU787
ALEU797
APEG807
AHOH905

site_idAC5
Number of Residues8
Detailsbinding site for residue EDO A 805
ChainResidue
ASER509
AHIS683
AMET687
AARG691
AGLN728
AHOH909
AHOH1053
AHOH1160

site_idAC6
Number of Residues6
Detailsbinding site for residue PEG A 806
ChainResidue
AASN457
AASP460
AHIS463
AARG520
ASER531
APHE533

site_idAC7
Number of Residues9
Detailsbinding site for residue PEG A 807
ChainResidue
ALYS512
ASER513
APRO688
AARG691
ASER796
AEDO804
AHOH905
AHOH980
AHOH1106

site_idAC8
Number of Residues4
Detailsbinding site for residue SCN A 808
ChainResidue
ATRP459
ATRP459
AASN523
AASN523

site_idAC9
Number of Residues7
Detailsbinding site for residue SCN A 809
ChainResidue
AGLN620
AGLU624
ALYS653
AGLY655
AASN663
AHOH981
AHOH1107

site_idAD1
Number of Residues4
Detailsbinding site for residue NA A 810
ChainResidue
AHOH972
AHOH1183
AHOH1220
AHOH1230

site_idAD2
Number of Residues4
Detailsbinding site for residue K A 811
ChainResidue
AHOH924
AHOH948
AHOH984
AHOH1245

site_idAD3
Number of Residues5
Detailsbinding site for residue GOL A 812
ChainResidue
AARG660
ATYR662
APHE793
ATRP794
AHOH920

site_idAD4
Number of Residues13
Detailsbinding site for residue N9W A 813
ChainResidue
ASER531
AHIS574
AGLY582
APHE583
AARG601
AASP612
AHIS614
APHE643
AASP705
AGLY743
ATYR745
AZN801
AHOH903

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PDB entries from 2024-06-26

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