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6TFB

Carbamazepine binds Frizzled8

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue GOL A 201
ChainResidue
ATHR39
AVAL40
APRO41
AGLN62
AASP63
AGLY66
AHOH303
BLEU159
BPHE160

site_idAC2
Number of Residues6
Detailsbinding site for residue GOL A 202
ChainResidue
ALEU33
ATYR52
ALEU97
ATYR100
ALYS101
ALYS102

site_idAC3
Number of Residues9
Detailsbinding site for residue N6W A 203
ChainResidue
AGLN56
ASER90
APRO94
APRO103
ALEU104
APRO105
AARG137
APRO139
AHOH329

site_idAC4
Number of Residues4
Detailsbinding site for residue GOL B 201
ChainResidue
APHE160
BTHR39
BGLN62
BASP63

site_idAC5
Number of Residues6
Detailsbinding site for residue N6W B 202
ChainResidue
BGLN56
BSER90
BPRO103
BLEU104
BPRO105
BHOH318

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues20
DetailsRegion: {"description":"Wnt-binding"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues14
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

244349

PDB entries from 2025-11-05

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