6SQ0
ERa_L536S (L536S/C381S/C471S,C530S) in complex with a bridged tetracyclic indole (compound 8)
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 9 |
Details | binding site for residue LRQ A 601 |
Chain | Residue |
A | LEU346 |
A | THR347 |
A | GLU353 |
A | LEU384 |
A | ARG394 |
A | PHE404 |
A | GLY521 |
A | HIS524 |
A | LEU525 |
site_id | AC2 |
Number of Residues | 10 |
Details | binding site for residue LRQ B 601 |
Chain | Residue |
B | MET343 |
B | LEU346 |
B | THR347 |
B | GLU353 |
B | LEU384 |
B | MET388 |
B | ARG394 |
B | PHE404 |
B | MET421 |
B | GLY521 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | MOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106 |
Chain | Residue | Details |
A | TYR537 | |
B | TYR537 |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | LIPID: S-palmitoyl cysteine => ECO:0000250 |
Chain | Residue | Details |
A | CYS447 | |
B | CYS447 |