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6PIT

Estrogen Receptor Alpha Ligand Binding Domain Y537S Mutant in Complex with SRC2 Stapled Peptide 41A and Estradiol

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue EST A 601
ChainResidue
ALEU346
AGLU353
ALEU387
AARG394
AMET421
AGLY521
AHIS524
ALEU525
AHOH736

site_idAC2
Number of Residues8
Detailsbinding site for residue EST B 601
ChainResidue
BMET343
BLEU346
BGLU353
BLEU387
BARG394
BMET421
BHIS524
BLEU525

site_idAC3
Number of Residues1
Detailsbinding site for Di-peptide ARG E 7 and LOU E 8
ChainResidue
CLEU9

site_idAC4
Number of Residues3
Detailsbinding site for Di-peptide LOU E 8 and LEU E 9
ChainResidue
AGLN375
AVAL376
CARG7

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsLipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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