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6O5Z

Crystal Structure of the human MLKL pseudokinase domain bound to compound 2

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues3
Detailsbinding site for residue EDO A 501
ChainResidue
AGLU250
AGLY349
AHOH631

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 502
ChainResidue
AALA228
AGLU284
ACYS286
ALEU338

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 503
ChainResidue
ATYR387
AGLU381
AASP384

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 504
ChainResidue
ATHR340
AGLY342
BTHR340
BGLY342
BGLN344

site_idAC5
Number of Residues17
Detailsbinding site for residue LN4 B 501
ChainResidue
BLEU209
BARG210
BLEU217
BALA228
BGLU250
BTHR253
BMET283
BGLU284
BTYR285
BCYS286
BGLU293
BHIS329
BLEU338
BLEU347
BALA348
BGLY349
BPHE350

site_idAC6
Number of Residues6
Detailsbinding site for residue EDO B 502
ChainResidue
BPRO379
BVAL424
BARG428
BGLN430
BARG449
BHIS451

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
ChainResidueDetails
ALEU209
BLEU209

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000305
ChainResidueDetails
ALYS230
BLYS230

site_idSWS_FT_FI3
Number of Residues2
DetailsMOD_RES: Phosphothreonine; by RIPK3 => ECO:0000269|PubMed:22265413
ChainResidueDetails
ATHR357
BTHR357

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: Phosphoserine; by RIPK3 => ECO:0000269|PubMed:22265413, ECO:0000269|PubMed:29883610
ChainResidueDetails
ASER358
BSER358

site_idSWS_FT_FI5
Number of Residues2
DetailsMOD_RES: Phosphoserine; by RIPK3 => ECO:0000250|UniProtKB:Q9D2Y4
ChainResidueDetails
ASER360
BSER360

220113

PDB entries from 2024-05-22

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