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6NWL

Structure of the Ancestral Glucocorticoid Receptor 2 ligand binding domain in complex with hydrocortisone and PGC1a coregulator fragment

Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue HCY A 301
ChainResidue
ALEU32
AVAL216
APHE218
AASN33
AGLN39
AARG80
APHE92
AGLN111
APHE204
ACYS205
ATHR208

site_idAC2
Number of Residues8
Detailsbinding site for residue GOL A 302
ChainResidue
AGLU9
AVAL12
ASER76
AARG80
ATYR132
AEPE305
AGOL307
AHOH447

site_idAC3
Number of Residues4
Detailsbinding site for residue GOL A 303
ChainResidue
ALYS83
AASN86
AASN86
AASN88

site_idAC4
Number of Residues10
Detailsbinding site for residue TLA A 304
ChainResidue
ATYR67
ASER68
ATRP69
AMET70
ASER71
ATHR143
AHIS195
AVAL198
ALEU202
AGLN229

site_idAC5
Number of Residues7
Detailsbinding site for residue EPE A 305
ChainResidue
AVAL12
ATRP79
AARG80
ALYS83
AGLN84
AGOL302
AHOH413

site_idAC6
Number of Residues1
Detailsbinding site for residue SCN A 306
ChainResidue
AARG159

site_idAC7
Number of Residues8
Detailsbinding site for residue GOL A 307
ChainResidue
AGLU9
APRO10
AALA43
ATRP46
ASER76
ALYS136
AGOL302
AHOH458

site_idAC8
Number of Residues6
Detailsbinding site for residue SCN A 308
ChainResidue
ALYS189
AASP192
AHIS244
AGLN245
ALYS246
AHOH462

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000250|UniProtKB:O70343
ChainResidueDetails
BLYS146

219140

PDB entries from 2024-05-01

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