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6MVY

NavAb voltage-gated sodium channel, residues 1-226, crystallized in the presence of Class 1B Anti-arrhythmic drug Lidocaine

Functional Information from GO Data
ChainGOidnamespacecontents
A0005216molecular_functionmonoatomic ion channel activity
A0005261molecular_functionmonoatomic cation channel activity
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0016020cellular_componentmembrane
A0055085biological_processtransmembrane transport
B0005216molecular_functionmonoatomic ion channel activity
B0005261molecular_functionmonoatomic cation channel activity
B0005886cellular_componentplasma membrane
B0006811biological_processmonoatomic ion transport
B0016020cellular_componentmembrane
B0055085biological_processtransmembrane transport
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue PX4 A 1301
ChainResidue
AILE1097
ALEU1151
APHE1152
ATYR1191
AALA1194
AHOH1418

site_idAC2
Number of Residues12
Detailsbinding site for residue PX4 A 1302
ChainResidue
APHE1167
ATYR1168
APHE1171
AMET1188
APRO1192
ATRP1195
AMET1209
APX41303
AHOH1413
AMET1137
AGLY1164
AGLU1165

site_idAC3
Number of Residues13
Detailsbinding site for residue PX4 A 1303
ChainResidue
AILE1022
AGLY1026
AILE1027
AGLY1030
ASER1034
ATHR1036
ALEU1109
ATHR1138
ATYR1142
ATHR1162
AGLY1164
APX41302
AHOH1402

site_idAC4
Number of Residues6
Detailsbinding site for residue PX4 A 1304
ChainResidue
APRO1075
ATRP1076
AVAL1120
ASER1121
AILE1124
ASER1125

site_idAC5
Number of Residues7
Detailsbinding site for residue SO4 A 1305
ChainResidue
APHE1156
APRO1157
AGLU1158
ATRP1159
AHOH1405
BSO41305
BHOH1402

site_idAC6
Number of Residues5
Detailsbinding site for residue PX4 B 1301
ChainResidue
BILE1097
BTYR1191
BTYR1193
BALA1194
BHOH1411

site_idAC7
Number of Residues11
Detailsbinding site for residue PX4 B 1302
ChainResidue
BMET1137
BGLY1164
BGLU1165
BPHE1167
BTYR1168
BPHE1171
BMET1188
BPRO1192
BTRP1195
BPX41303
BHOH1401

site_idAC8
Number of Residues12
Detailsbinding site for residue PX4 B 1303
ChainResidue
BILE1022
BGLY1026
BILE1027
BGLY1030
BSER1034
BTHR1138
BTYR1142
BTHR1162
BLEU1163
BGLY1164
BPX41302
BHOH1410

site_idAC9
Number of Residues3
Detailsbinding site for residue PX4 B 1304
ChainResidue
BTRP1076
BSER1121
BILE1124

site_idAD1
Number of Residues7
Detailsbinding site for residue SO4 B 1305
ChainResidue
ASO41305
AHOH1405
BPHE1156
BPRO1157
BGLU1158
BTRP1159
BHOH1402

221051

PDB entries from 2024-06-12

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