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6MF9

Crystal structure of CGD4-650 with compound BI2536

Functional Information from GO Data
ChainGOidnamespacecontents
A0000124cellular_componentSAGA complex
A0046695cellular_componentSLIK (SAGA-like) complex
B0000124cellular_componentSAGA complex
B0046695cellular_componentSLIK (SAGA-like) complex
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue R78 A 3000
ChainResidue
AVAL1871
AILE1880
AALA1881
ATYR1926
AASN1927
AHOH3117
BASN1883
BILE1925
BTYR1926

site_idAC2
Number of Residues11
Detailsbinding site for residue R78 B 3000
ChainResidue
AASN1883
AILE1925
ATYR1926
BVAL1871
BVAL1876
BILE1880
BALA1881
BTYR1926
BASN1927
BLEU1933
BHOH3110

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. ShvFwnrvSeriap..NYYnlVkrpMwlqlMinkckkre..Yksrkdfqddldl.IveNCkiY
ChainResidueDetails
ASER1869-TYR1926

226262

PDB entries from 2024-10-16

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