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6M8Q

Cleavage and Polyadenylation Specificity Factor Subunit 3 (CPSF3) in complex with NVP-LTM531

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue ZN A 501
ChainResidue
AASP75
AHIS76
AASP179
AHIS418
AZN502
APO4505
AHOH630

site_idAC2
Number of Residues7
Detailsbinding site for residue ZN A 502
ChainResidue
AHIS158
AASP179
AZN501
APO4505
AHOH630
AHIS71
AHIS73

site_idAC3
Number of Residues19
Detailsbinding site for residue JBG A 503
ChainResidue
AILE43
AHIS44
APRO45
ALEU47
AGLU48
AALA52
ATYR110
APRO239
AVAL240
APHE241
APRO329
AGLY330
AMET331
AGLN333
AGLY356
AHOH637
AHOH647
AHOH663
AHOH672

site_idAC4
Number of Residues7
Detailsbinding site for residue PO4 A 504
ChainResidue
ATYR207
AHIS212
AGLU213
AARG218
ASER392
AHOH714
BARG426

site_idAC5
Number of Residues12
Detailsbinding site for residue PO4 A 505
ChainResidue
AHIS73
AASP75
AHIS158
AASP179
ATYR357
AHIS396
AHIS418
AZN501
AZN502
AHOH608
AHOH630
AHOH671

site_idAC6
Number of Residues7
Detailsbinding site for residue ZN B 501
ChainResidue
BASP75
BHIS76
BASP179
BHIS418
BZN502
BPO4504
BHOH603

site_idAC7
Number of Residues7
Detailsbinding site for residue ZN B 502
ChainResidue
BHIS71
BHIS73
BHIS158
BASP179
BZN501
BPO4504
BHOH603

site_idAC8
Number of Residues17
Detailsbinding site for residue JBG B 503
ChainResidue
BILE43
BHIS44
BPRO45
BLEU47
BLEU74
BTYR110
BSER114
BPRO239
BVAL240
BPHE241
BPRO329
BGLY330
BMET331
BGLY356
BHOH637
BHOH641
BHOH683

site_idAC9
Number of Residues13
Detailsbinding site for residue PO4 B 504
ChainResidue
BHIS73
BASP75
BHIS158
BASP179
BTYR357
BSER394
BHIS396
BHIS418
BZN501
BZN502
BHOH603
BHOH618
BHOH674

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Proton donor => ECO:0000255
ChainResidueDetails
AHIS396
BHIS396

site_idSWS_FT_FI2
Number of Residues14
DetailsBINDING: BINDING => ECO:0000269|PubMed:17128255, ECO:0007744|PDB:2I7T, ECO:0007744|PDB:2I7V
ChainResidueDetails
AHIS71
BASP75
BHIS76
BHIS158
BASP179
BHIS418
AHIS73
AASP75
AHIS76
AHIS158
AASP179
AHIS418
BHIS71
BHIS73

site_idSWS_FT_FI3
Number of Residues2
DetailsMOD_RES: N-acetylserine => ECO:0007744|PubMed:19413330, ECO:0007744|PubMed:22223895
ChainResidueDetails
ASER2
BSER2

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PDB entries from 2024-07-31

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