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6G05

RORGT (264-518;C455S) IN COMPLEX WITH INVERSE AGONIST "CPD-2" AND RIP140 PEPTIDE AT 1.90A

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue EF5 A 601
ChainResidue
ACYS285
AALA368
APHE377
APHE378
APHE388
AILE400
APHE401
AHOH710
AHOH749
AGLN286
ALEU287
ACYS320
AHIS323
ALEU324
AARG364
AMET365
AARG367

site_idAC2
Number of Residues17
Detailsbinding site for residue EF5 B 601
ChainResidue
BCYS285
BGLN286
BLEU287
BCYS320
BHIS323
BLEU324
BARG364
BMET365
BARG367
BALA368
BPHE377
BPHE378
BPHE388
BILE400
BPHE401
BHOH708
BHOH741

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
PLYS508
QLYS508

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PDB entries from 2024-07-17

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