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6FYM

Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor ITK1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ ADP-ribosyltransferase activity
D0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue EBB A 1901
ChainResidue
AHIS1682
ALEU1782
DTHR1726
AGLY1683
ATHR1684
AASP1685
ATYR1701
AGLY1703
ATYR1714
ATYR1721
ATYR1727

site_idAC2
Number of Residues10
Detailsbinding site for residue EBB B 1901
ChainResidue
BHIS1682
BGLY1683
BTHR1684
BASP1685
BTYR1701
BGLY1703
BTYR1714
BSER1722
BTYR1727
CTHR1726

site_idAC3
Number of Residues8
Detailsbinding site for residue EBB C 1901
ChainResidue
BTHR1726
CHIS1682
CGLY1683
CASP1685
CTYR1714
CTYR1721
CSER1722
CTYR1727

site_idAC4
Number of Residues3
Detailsbinding site for residue NO3 C 1902
ChainResidue
BTYR1721
CTYR1709
CTYR1721

site_idAC5
Number of Residues13
Detailsbinding site for residue EBB D 1901
ChainResidue
ATHR1726
DHIS1682
DGLY1683
DTHR1684
DASP1685
DTYR1701
DGLY1703
DTYR1714
DTYR1721
DSER1722
DTYR1727
DLEU1782
DNO31902

site_idAC6
Number of Residues4
Detailsbinding site for residue NO3 D 1902
ChainResidue
AALA1708
DTYR1721
DTYR1727
DEBB1901

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PDB entries from 2024-07-10

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